V. Finger, T. Kucera, R. Kafkova, L. Muckova, R. Dolezal, J. Kubes, M. Novak, L. Prchal, L. Lakatos, M. Andrs, M. Hympanova, J. Marek, M. Kufa, V. Spiwok, O. Soukup, E. Mezeiova, J. Janousek, L. Nevosadova, M. Benkova, R.R.A. Kitson, M. Kratky, S. Bősze, K. Mikusova, R. Hartkoorn, J. Roh, J. Korabecny, 2,6-Disubstituted 7-(naphthalen-2-ylmethyl)-7H-purines as a new class of potent antitubercular agents inhibiting DprE1, Eur. J. Med. Chem. 2023, 258, 115611. (IF2022 = 6.7) (QAIS1)
N. Monakhova, J. Kordulakova, A. Vocat, A. Egorova, A. Lepioshkin, E. G. Salina, J. Nosek, E. Repkova, J. Zemanova, H. Jurdakova, R. Gorova, J. Roh, G. Degiacomi, J. C. Sammartino, M. R. Pasca, S. T. Cole, K. Mikusova, V. Makarov. Design and Synthesis of Pyrano[3,2-b]indolones Showing Antimycobacterial Activity.ACS Infect. Dis. 2021, 7(1), 88-100. (IF2019 = 5.084) (DAIS1)
Krátký M., Konečná K., Brokešová K., Maixnerová J., Trejtnar F., Vinšová J. Optimizing the structure of (salicylideneamino)benzoic acids: Towards selective antifungal and anti-staphylococcal agents, Eur. J. Pharm. Sci. 2021, 159, 105732 [ISSN 0928-0987, IF2019 = 3.616]. https://doi.org.10.1016/j.ejps.2021.105732
Y.Sheena Mary, Y.Shyma Mary, Krátký M., Vinsova J., Baraldi C., Gamberini M.C. Concentration dependent SERS, DFT and molecular docking studies of a ureido derivative with antitubercular properties. Spectrochim. Acta A2021, 249, 119329 [ISSN 1386-1425, IF2019= 3.232]. https://doi.org/10.1016/j.saa.2020.119329
Y. Sheena Mary, Y. Shyma Mary, Krátký M., Vinsova J., Baraldi C., Gamberini M.C. DFT, SERS-concentration and solvent dependent and docking studies of a bioactive benzenesulfonamide derivative. J. Mol. Struct.2021, 1228 129680. [ISSN 0022-2860, IF2019 = 2.463]. https://doi.org/10.1016/j.molstruc.2020.129680
Gamberinia M. C., Y.Shyma Mary, Y.Sheena Mary, Krátký M., Vinsova J., Baraldi C. Spectroscopic investigations, concentration dependent SERS, and molecular docking studies of a benzoic acid derivative. Spectrochim. Acta A2021, 248, 119265 [ISSN 1386-1425, IF2019= 3.232]. https://doi.org/10.1016/j.saa.2020.119265
Krátký M., Baranyai Z., Štěpánková Š., Svrčková K., Švarcová M., Stolaříková J., Horváth L., Bősze S., Vinšová J. N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1- carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity. Molecules2020, 25, 2268; https.//doi.org/10.3390/molecules25102268. [ISSN 1420-3049, IF2019 = 3.267].
Ambrożkiewicz W., Kučerová-Chlupáčová M., Janďourek O., Konečná K., Paterová P., Bárta P., Vinšová J., Doležal M., Zitko J. 5-Alkylamino-N-Phenylpyrazine-2-Carboxamides: Design, Preparation, And Antimycobacterial Evaluation. Molecules2020, 25, 1561; https://doi.org/10.3390/molecules25071561 [ISSN 1420-3049, IF2019 = 3.267].
Krátký M., Konečná K., Janoušek J., Brablíková M., Janďourek O., Trejtnar F., Stolaříková J., Vinšová J. 4-Aminobenzoic acid derivatives: Converting folate precursor to antimicrobial and cytotoxic agents. Biomolecules 2020, 10, 9, 1-21. doi:10.3390/biom10010009. [IF2019= 4,082].
Krátký M., Jaklová K., Štěpánková Š., Svrčková K., Pflégr V., Vinšová J. N-[3,5-Bis(trifluoromethyl)phenyl]-5-bromo-2-hydroxybenzamide Analogues: Novel Acetyl- and Butyrylcholinesterase Inhibitors. Curr. Top. Med. Chem. 2020, 20(23), 2094-2105. https://doi.org/10.2174/1568026620666200819154722 [IF2019 = 3,218]
Krátký M., Štěpánková Š., Brablíková M., Svrčková K. Švarcová M., Vinšová J. Novel Iodinated Hydrazide-hydrazones and their Analogues as Acetyl- and Butyrylcholinesterase Inhibitors. Curr. Top. Med. Chem. 2020, 20, (23), 2106-2117. https://doi.org/10.2174/1568026620666200819155503 [IF2019 = 3,218].
Krátký M., Štěpánková Š., Houngbedji Neto-Honorius, Vosátka R., Vorčáková K., Vinšová J. 2-Hydroxy-N-phenylbenzamides and their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase. Biomolecules 2019, 9, 698; doi:10.3390/biom9110698, [IF2019= 4,082]]
Krátký M., Janďourek O., Baranyai Zs., Novotná E., Stolaříková J., Bősze S., Vinšová J. Phenolic N-monosubstituted carbamates: Antitubercular and toxicity evaluation of multi-targeting compounds. Eur. J. Med. Chem. 2019, 181, 111578 [ISSN 0223-5234, IF2019= 5.572].
Krátký M., Vorčáková K., Vinšová J., Štěpánková Š. Investigation of salicylanilide and 4-chlorophenol-based N-monosubstituted carbamates as potential inhibitors of acetyl- and butyrylcholinesterase, Bioorg. Chem.2018, 80, 668-673 [ISSN 0968-0896, IF2017 = 3.929].
Zitko J., Janďourek O., Paterová P., Navrátilová L., Kuneš J., Vinšová J., Doležal M. Design, synthesis and antimycobacterial activity of hybrid molecules combining pyrazinamide with 4-phenylthiazol-2-amine scaffold. MedChemComm.2018. 9(4), 685-696. [ISSN 2040-2503], IF2017 = 2.342, doi: http://dx.doi.org/10.1039/C8MD00056E
Pospíšilová Š., Michnová H., Pauk K., Vinšová J., Imramovský A., Čížek A., Jampílek J. In vitro activity of salicylamide derivatives against vancomycin-resistant enterococci. Bioorg. Med. Chem. Letters2018, 28, 2184-2188. [ISSN 0960-894X, IF2017 = 2.442]
Vosátka R., Krátký M., Švarcová M., Janoušek J., Stolaříková J., Madacki J., Husza S., Mikušová K., Korduláková J.,Trejtnar F., Vinšová J. New lipophilic isoniazid derivatives and their 1,3,4-oxadiazole analogues: Synthesis, antimycobacterial activity and investigation of their mechanism of action. Eur. J. Med. Chem. 2018,151, 824-835. [ISSN 0223-5234, IF2017 = 4,816]
Vosátka R., Krátký M., Vinšová J. Triclosan and its derivatives as antimycobacterial active agents Eur. J. Pharm. Sci. 2018, 114, 318–331. [ISSN 0928-0987, IF2016 = 3.466]. doi.org/10.1016/j.ejps.2017.12.013
Krátký M., Bősze S., Baranyai Zs., Stolaříková J., Vinšová J. Synthesis and biological evolution of hydrazones derived from 4-(trifluoromethyl)benzohydrazide. Bioorg. Med. Chem. Lett.2017, 27,5185-5189. [ISSN 0960-894X, IF2016 = 2.454]. doi: 10.1016/j.bmcl.2017.10.050
Krátký M., Dzurková M., Janoušek O., Konečná K., Trejtnar F., Stolaříková J., Vinšová J. Sulfadiazine Salicylaldehyde-Based Schiff Bases: Synthesis, Antimicrobial Activity and Cytotoxicity. Molecules2017, 22, 1573 [ISSN 1420-3049, IF2016 = 2.861]. doi:10.3390/molecules22091573
Krátký M., Stolaříková J., Vinšová J. Antimicrobial activity of rhodanine-3-acetic acid derivatives. Bioorg. Med. Chem. 2017, 25(6), 1839–1845 [ISSN 0968-0896, IF2016 = 2.930]. https://doi.org/10.1016/j.bmc.2017.01.045
Baranyai Zs, Krátký M., Vosátka M., Szabó N., Senoner Sz., Dávid S., Stolaříková J., Vinšová J., Bősze S. In vitro biological evaluation of new antimycobacterial salicylanilide-tuftsin conjugates. Europ. J. Med. Chem. 2017, 133, 152-173 [ISSN 0223-5234, IF2016 = 4.519]. https://doi.org/10.1016/j.ejmech.2017.03.047
Krátký M., Stolaříková J., Vinšová J. Novel Sulfamethoxazole Ureas and Oxalamides as Potential Antimicobacterial Agents. Molecules2017, 22(4), 535 [ISSN 1420-3049, IF2016 = 2.861]. doi:10.3390/molecules22040535
Krátký M., Vinšová J., Štěpánková Š., Vorčáková K., Navrátilová L., Trejtnar F., Stolaříková J. Novel Fluorophenylalanine Derivatives: Synthesis and Investigation of Their Biological Activity. Bioorganic Chemistry 2017, 71, 244 - 256 [ISSN: 0045-2068, IF2016 = 3.402]. https://doi.org/10.1016/j.bioorg.2017.02.010
Paraskevopoulos G., Monteiro S., Vosátka R., Krátký M., Navrátilová L., Trejtnar F., Stolaříková J., Vinšová J. Novel salicylanilides from 4,5-dihalogenated salicylic acids: Synthesis, antimicrobial activity and cytotoxicity. Bioorg. Med. Chem. 2017, 25(4), 1524-1532 [ISSN 0968-0896, IF2016 = 2.930]. http://dx.doi.org/10.1016/j.bmc.2017.01.016
Krátký M., Štěpánková Š., Vorčáková K., Vinšová J. Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors. Bioorganic Chemistry 2016, 68, 23-29 [ISSN 0045-2068, IF2016 = 3.231].
Krátký M., Vinšová J. Salicylanilide N-monosubstituted carbamates: Synthesis and in vitro antimicrobial activity. Bioorg. Med. Chem. 2016, 24(6), 1322-1330. http://dx.doi.org/10.1016/j.bmc.2016.02.004 [ISSN 0968-0896, IF20156= 2.930].
Krátký M., Štěpánková Š., Vorčáková K., Švarcová M, Vinšová J. Novel Cholinesterases Inhibitors Based on O-Aromatic N,N-Disubstituted Carbamates and Thiocarbamate, Molecules, 2016, 21, 191-201. [ISSN 1420-3049, IF2016 = 2.861].
Krátký M., Vinšová J. Sulphur-Containing Heterocycles as Antimycobacterial Agents: Recent Advances in Thiophene and Thiadiazole Derivatives, Current Topics in Medicinal Chemistry, 2016, 16(26), 2921-2952 [ISSN 1389-4501, IF2016 = 2.561]. DOI: 10.2174/1568026616666160506131118