Selected publications

Publications - since 2010

 

Development of new potential drugs with antimicrobial activity

2018

  • Vosátka R., Krátký M., Vinšová J. Triclosan and its derivatives as antimycobacterial active agents Eur. J. Pharm. Sci. 2018, 114, 318–331. [ISSN 0928-0987, IF2016 = 3.756]. doi.org/10.1016/j.ejps.2017.12.013

2017

  • Krátký M., Bősze S., Baranyai Zs., Stolaříková J., Vinšová J. Synthesis and biological evolution of hydrazones derived from 4-(trifluoromethyl)benzohydrazide. Bioorg. Med. Chem. Lett. 2017, 27,5185-5189. [ISSN 0960-894X, IF2016 = 2.454]. doi: 10.1016/j.bmcl.2017.10.050
  • Krátký M., Dzurková M., Janoušek O., Konečná K., Trejtnar F., Stolaříková J., Vinšová J. Sulfadiazine Salicylaldehyde-Based Schiff Bases: Synthesis, Antimicrobial Activity and Cytotoxicity. Molecules 2017, 22, 1573 [ISSN 1420-3049, IF2016 = 2.861]. doi:10.3390/molecules22091573
  • Krátký M., Stolaříková J., Vinšová J. Antimicrobial activity of rhodanine-3-acetic acid derivatives. Bioorg. Med. Chem. 2017, 25(6), 1839–1845 [ISSN 0968-0896, IF2016 = 2.930]. https://doi.org/10.1016/j.bmc.2017.01.045
  • Baranyai Zs, Krátký M., Vosátka M., Szabó N., Senoner Sz., Dávid S., Stolaříková J., Vinšová J., Bősze S. In vitro biological evaluation of new antimycobacterial salicylanilide-tuftsin conjugates. Europ. J. Med. Chem. 2017, 133, 152-173 [ISSN 0223-5234, IF2016 = 4.519]. https://doi.org/10.1016/j.ejmech.2017.03.047
  • Krátký M., Stolaříková J., Vinšová J. Novel Sulfamethoxazole Ureas and Oxalamides as Potential Antimicobacterial Agents. Molecules 2017, 22(4), 535 [ISSN 1420-3049, IF2016 = 2.861]. doi:10.3390/molecules22040535
  • Krátký M., Vinšová J., Štěpánková Š., Vorčáková K., Navrátilová L., Trejtnar F., Stolaříková J. Novel Fluorophenylalanine Derivatives: Synthesis and Investigation of Their Biological Activity. Bioorganic Chemistry 2017, 71, 244 - 256 [ISSN: 0045-2068, IF2016 = 3.402]. https://doi.org/10.1016/j.bioorg.2017.02.010
  • Paraskevopoulos G., Monteiro S., Vosátka R., Krátký M., Navrátilová L., Trejtnar F., Stolaříková J., Vinšová J. Novel salicylanilides from 4,5-dihalogenated salicylic acids: Synthesis, antimicrobial activity and cytotoxicity. Bioorg. Med. Chem. 2017, 25(4), 1524-1532 [ISSN 0968-0896, IF2016 = 2.930]. http://dx.doi.org/10.1016/j.bmc.2017.01.016 

2016

  • Krátký M.*, Štěpánková Š., Vorčáková K., Vinšová J. Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors. Bioorganic Chemistry 2016, 68, 23-29  [ISSN 0045-2068, IF2016 = 3.231].
  • Kozic J.*, Novák Z., Římal V., Profant V., Kuneš J., Vinšová J. Conformations, equilibrium thermodynamics and rotational barriers of secondary thiobenzanilides. Tetrahedron, 2016, 72, 2072-2083 [ISSN: 0040-4020, IF2016 = 2.651]. doi:10.1016/j.tet.2016.02.035
  • Krátký M.*, Vinšová J. Salicylanilide N-monosubstituted carbamates: Synthesis and in vitro antimicrobial activity. Bioorg. Med. Chem. 201624(6), 1322-1330. http://dx.doi.org/10.1016/j.bmc.2016.02.004   [ISSN 0968-0896, IF20156= 2.930].
  • Krátký M.*, Štěpánková Š., Vorčáková K., Švarcová M, Vinšová J. Novel Cholinesterases Inhibitors Based on O-Aromatic N,N-Disubstituted Carbamates and Thiocarbamate, Molecules, 201621, 191-201. [ISSN 1420-3049, IF2016 = 2.861].
  • Krátký M.*, Vinšová J. Sulphur-Containing Heterocycles as Antimycobacterial Agents: Recent Advances in Thiophene and Thiadiazole Derivatives, Current Topics in Medicinal Chemistry, 201616(26), 2921-2952 [ISSN 1389-4501, IF2016 = 2.561]. DOI: 10.2174/1568026616666160506131118

2015

  • Krátký M., Štěpánková Š, Vorčáková K., Vinšová J.* Salicylanilide Diethyl Phosphates as Cholinesterases Inhibitors. Bioorg. Med. Chem. 2015, 58, 48-52. [ISSN 0968-0896, IF2015 = 2.923].
  • Zadrazilova I., Pospisilova S., Pauk K., Imramovsky A., Vinsova J., Cizek A., Jampilek J.* In vitro bactericidal activity of 4- and 5-chloro-2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides against MRSA, BioMed Research International, 2015 Article 349534[ISSN 2314-6133, IF2014 = 1.579].
  • Krátký M., Bősze S., Baranyai Zs., Szabó I., Stolaříková J., Paraskevopoulos G., Vinšová J.* Synthesis and In Vitro Biological Evaluation of 2-(Phenylcarbamoyl)phenyl 4-Substituted Benzoates. Bioorg. Med. Chem. 201524(4), 868–875.  [ISSN 0968-0896, IF2015 = 2.793].
  • Švarcová M., Krátký M., Vinšová J*. Investigation of potential inhibitors of chorismate-utilizing enzymes Curr. Med. Chem. 2015, 22(11), 1383-1399 [ISSN 0929-8673, IF2015 = 3.853].
  • Krátký M.*, Mandíková J., Trejtnar F., Buchta V., Stolaříková J., Vinšová J. Synthesis and antimicrobial activity of novel sulfamethoxazole ureas and 2,4,5- imidazolidin-2,4,5-triones. Chemical Papers,  2015, 69(8), 1108-1117. [ISSN 0366-6352, IF2015 = 1.326].
  • Zadrazilova I., Masarikova M., Pospisilova S., Imramovsky A., Ferriz J.M., Vinsova J., Cizek J., Jampilek J.* Salicylanilide carbamates: Promising antibacterial agents with high in vitro activity against methicillin-resistant Staphylococcus aureus (MRSA), Eur. J. Pharm. Sci., 2015, 77, 197-207. [ISSN 0928-0987, IF2015 = 3.350].
  • Baranyai Z., Krátký M., Vinšová J., Szabó N., Senoner Z., Horváti K., Stolaříková J., Dávid S., Bősze S.* Combating highly resistant emerging pathogen Mycobacterium abscessus and Mycobacterium tuberculosis with novel salicylanilide esters and carbamates. Europ. J. Med. Chem. 2015101, 692-704. [ISSN 0223-5234, IF2015 = 3.447].
  • Paraskevopoulos G., Krátký M., Mandíková J., Trejtnar F., Stolaříková J., Pávek P., Besra G.,Vinšová J.* Novel derivatives of nitro-substituted salicylic acids: Synthesis, antimicrobial activity and cytotoxicity. Bioorg. Med. Chem. 2015, 23, 7292-7301 [ISSN 0968-0896, IF2015 = 2.923].

2014

2013

2012

2011

2010

 

Development of new antituberculosis drugs

2017

2016

2015

2014

2013

2012

2010

 

Synthesis of dexrazoxane analogues and iron chelators

2018

2017

2016

2015

2014

© Charles University, Faculty of Pharmacy in Hradec Králové, Akademika Heyrovského 1203, 500 05 Hradec Králové, Czech Republic
Website information | Powered by Kentico