2020
Nawrot D., Suchánková E., Janďourek O., Konečná K., Bárta P., Doležal M., Zitko J. 2020. N-pyridinylbenzamides: an isosteric approach towards new antimycobacterial compounds, Chem Biol Drug Des.https://doi.org/10.1111/cbdd.13804. IF[2019]= 2.548
Juhás M., Kučerová L., Horáček O., Janďourek O., Kubíček V., Konečná K., Kučera R., Bárta P., Janoušek J., Paterová P., Kuneš J., Doležal M., Zitko J. 2020. N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents-the Synthesis and Biological Evaluation of Enantiomers. Molecules. 25(7):1518. https://doi.org/10.3390/molecules25071518. IF[2019]= 3.267
Ambrożkiewicz W., Kučerová-Chlupáčová M., Janďourek O., Konečná K., Paterová P., Bárta P., Vinšová J., Doležal M., Zitko J. 2020. 5-Alkylamino-N-phenylpyrazine-2-carboxamides: Design, Preparation, and Antimycobacterial Evaluation. Molecules. 25(7):1561. https://doi.org/10.3390/molecules25071561. IF[2019]= 3.267
Bouz G., Juhás M., Pausas Otero L., Paredes de la Red C., Janďourek O., Konečná K., Paterová P., Kubíček V., Janoušek J., Doležal M., Zitko J. 2020. Substituted N-(Pyrazin-2-yl)benzenesulfonamides; Synthesis, Anti-Infective Evaluation, Cytotoxicity, and In Silico Studies. Molecules. 25(1):138. https://doi.org/10.3390/molecules25010138. IF[2019]=3.267
Krátký M., Konečná K., Janoušek J., Brablíková M., Janďourek O., Trejtnar F., Stolaříková J., Vinšová J. 2020. 4-Aminobenzoic Acid Derivatives: Converting Folate Precursor to Antimicrobial and Cytotoxic Agents. Biomolecules. 10(1):9. https://doi.org/10.3390/biom10010009 . IF[2019]= 4.082
2019
Konečná K., Klimentová J., Benada O., Němečková I., Janďourek O., Jílek P., Vejsová M. 2019. A comparative analysis of protein virulence factors released via extracellular vesicles in two Candida albicans strains cultivated in a nutrient-limited medium.
Microb Pathog. 136:103666. https://doi.org/10.1016/j.micpath.2019.103666. IF[2018]= 2.581
Karabanovich G., Dušek J., Savková K., Pavliš O., Pávková I., Korábečný J., Kučera T., Kočová Vlčková H., Huszár S., Konyariková Z., Konečná K., Janďourek O., Stolaříková J., Korduláková J., Vávrová K., Pávek P., Klimešová V., Hrabálek A., Mikušová K., Roh J. 2019. Development of 3,5-Dinitrophenyl-Containing 1,2,4-Triazoles and Their Trifluoromethyl Analogues as Highly Efficient Antitubercular Agents Inhibiting Decaprenylphosphoryl-beta-D-ribofuranose 2 '-Oxidase. J Med Chem. 62(17):8115-8139. https://doi.org/10.1021/acs.jmedchem.9b00912 . IF[2019]= 6.205
Krátký M., Janďourek O., Baranyai Z., Novotná E., Stolaříková J., Bősze S., Vinšová J. 2019. Phenolic N-monosubstituted Chem carbamates: Antitubercular and toxicity evaluation of multi-targeting compounds. Eur. J. Med Chem.181, 111578. https://doi.org/10.1016/j.ejmech.2019.111578 . IF[2019]= 5.573
Bouz G., Semelková L., Janďourek O., Konečná K., Paterová P., Navrátilová L., Kubíček V., Kuneš J., Doležal M., Zitko J. 2019. Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity.
Molecules. 24(7):1212. https://doi.org/10.3390/molecules24071212 . IF[2019]= 3,267
2018
Zitko J., Janďourek O., Paterová P., Navrátilová L., Kuneš J., Vinšová J., Doležal M. 2018. Design, synthesis and antimycobacterial activity of hybrid molecules combining pyrazinamide with a 4-phenylthiazol-2-amine scaffold. Med Chem Comm. 9, 685-696. https://doi.org/10.1039/C8MD00056E .
IF[2018]= 2.410
Zitko J., Mindlová A., Valášek O., Jand'ourek O., Paterová P., Janoušek J., Konečná K., Doležal M. Design, Synthesis and Evaluation of N-pyrazinylbenzamides as Potential Antimycobacterial Agents. 2018. Molecules. 23(9):2390. https://doi.org/10.3390/molecules23092390 . IF[2018]= 3.060
Horký P., Voráčová M., Konečná K., Sedlák D., Bartůněk P., Vacek J., Kuneš J., Pour M. 2018. Nontoxic combretafuranone analogues with high in vitro antibacterial activity. Eur J Med Chem. 143:843-853. https://doi.org/10.1016/j.ejmech.2017.11.078 . IF[2018]= 4.883
2017
Semelková L., Janošcová P., Fernandes C., Bouz G., Janďourek O., Konečná K., Paterová P., Navrátilová L., Kuneš J., Doležal M., Zitko J. 2017. Design, Synthesis, Antimycobacterial Evaluation, and In Silico Studies of 3-(Phenylcarbamoyl)-pyrazine-2-carboxylic Acids.
Molecules. 22(9):1491. https://doi.org/10.3390/molecules22091491 . IF[2017]= 3.098
Bouz G., Juhás M., Niklová P., Janďourek O., Paterová P., Janoušek J., Tůmová L., Kovalíková Z., Kastner P., Doležal M., Zitko J. 2017. Ureidopyrazine Derivatives: Synthesis and Biological Evaluation as Anti-Infectives and Abiotic Elicitors. Molecules. 22, 1797. https://doi.org/10.3390/molecules22101797 . IF[2017]= 3.098
Krátký M., Dzurková M., Janoušek J., Konečná K., Trejtnar F., Stolaříková J., Vinšová J. 2017. Sulfadiazine Salicylaldehyde-Based Schiff Bases: Synthesis, Antimicrobial Activity and Cytotoxicity. Molecules. 22(9):1573. https://doi.org/10.3390/molecules22091573 . IF[2017]= 3.098
Špaček J., Kestřánek J., Jílek P., Leško D., Plucnarová S., Buchta V. 2017. Comparison of two long-term gestagen regimens in the management of recurrent vulvovaginal candidiasis: A pilot study. Mycoses. 60(4):260-265. https://doi.org/10.1111/myc.12593 . IF[2017]= 2.793
Leško D., Buchta V., Salavec M., Jílek P., Kestřánek J., Drbohlavová A., Špaček J. 2017. Contemporary technicqes in diagnostic patients with vaginal microbiota. Ceska Gynekol. 82(2):152-157.
Němeček J., Sychra P., Macháček M., Benková M., Karabanovich G., Konečná K., Kavková V., Stolaříková J., Hrabálek A., Vávrová K., Soukup O., Roh J., Klimešová V. 2017. Structure-activity relationship studies on 3,5-dinitrophenyl tetrazoles as antitubercular agents. Eur J Med Chem. 130:419-432. https://doi.org/10.1016/j.ejmech.2017.02.058 . IF[2017]= 4.816
Semelková L., Janďourek O., Konečná K., Paterová P., Navrátilová L., Trejtnar F., Kubíček V., Kuneš J., Doležal M., Zitko J. 2017. 3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation. Molecules. 22(3):495. https://doi.org/10.1016/j.ejmech.2017.02.058 . IF[2017]= 3.098
Janďourek O., Tauchman M., Paterová P., Konečná K., Navrátilová L., Kubíček V., Holas O., Zitko J., Doležal M. 2017. Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation. Molecules. 22(2):223. https://doi.org/10.3390/molecules22020223 . IF[2017]= 3.098
Karabanovich G., Němeček J., Valášková L., Carazo A., Konečná K., Stolaříková J., Hrabálek A., Pavliš O., Pávek P., Vávrová K., Roh J., Klimešová V. 2017. S-substituted 3,5-dinitrophenyl 1,3,4-oxadiazole-2-thiols and tetrazole-5-thiols as highly efficient antitubercular agents. Eur J Med Chem. 126:369-383. https://doi.org/10.1016/j.ejmech.2016.11.041. IF[2017]= 4.816
2016
Kučerová-Chlupáčová M., Vyškovská-Tyllová V., Richterová-Finková L., Kuneš J., Buchta V., Vejsová M., Paterová P., Semelková L., Janďourek O., Opletalová V. 2016. Novel halogenated pyrazine-based chalcones as potential antimicrobial drugs. Molecules. 21, 1421. https://doi.org/10.3390/molecules21111421 . IF[2016]= 2.861
Karabanovich G., Zemanová J., Smutný T., Székely R., Šarkan M., Centárová I., Vocat A., Pávková I., Čonka P., Němeček J., Stolaříková J., Vejsová M., Vávrová K., Klimešová V., Hrabálek A., Pávek P., Cole ST., Mikušová K., Roh J. 2016. Development of 3,5-Dinitrobenzylsulfanyl-1,3,4-oxadiazoles and Thiadiazoles as Selective Antitubercular Agents Active Against Replicating and Nonreplicating Mycobacterium tuberculosis. J Med Chem. 59(6):2362-80.https://doi.org/10.1021/acs.jmedchem.5b00608 . IF[2016]= 6.256
Opletalová V., Doležel J., Kuneš J., Buchta V., Vejsová M., Kučerová-Chlupáčová M. 2016. Synthesis and Antifungal Screening of 2-{[1-(5-Alkyl/arylalkylpyrazin-2-yl)ethylidene]hydrazono}-1,3-thiazolidin-4-ones. Molecules. 21(11):1592. https://doi.org/10.3390/molecules21111592 . IF[2016]= 2.861
2015
Semelková L., Konečná K., Paterová. P, Kubíček V., Kuneš J., Nováková L., Marek J., Naesens L., Pesko M., Králová K., Doležal M., Zitko J. 2015. Synthesis and Biological Evaluation of N-Alkyl-3-(alkylamino)-pyrazine-2-carboxamides. Molecules. 20(5):8687-711. https://doi.org/10.3390/molecules21111421 . IF[2015]= 2.465
Servusová-Vaňásková B., Janďourek O., Paterová P., Korduláková J., Pleváková M., Kubíček V., Kučera R., Garaj V., Naesens L., Kuneš J., Doležal M., Zitko J. 2015. Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: Synthesis and antimycobacterial evaluation. Med. Chem. Comm. 6, 1311-1317. doi: 10.1039/c5md00178a . IF[2015]= 2.54
Janďourek O., Kuneš J., Doležal M. 2015. Microwave-Assisted Synthesis of Pyrazinamide Derivatives: the Coupling Reaction of 3-Chloropyrazine-2-Carboxamide and Ring-Substituted Anilines. Curr. Org. Synthesis.12, 189-196. https://doi.org/10.2174/1570179411999141106101501 . IF[2015]= 2.227
Zitko J., Servusová B., Janoutová A., Paterová P., Mandíková J., Garaj V., Vejsová M., Marek J., Doležal M. 2015. Synthesis and antimycobacterial evaluation of 5-alkylamino-N-phenylpyrazine-2-carboxamides. Bioorg Med Chem. 2015 Jan 1;23(1):174-83. https://doi.org/10.1016/j.bmc.2014.11.014 . IF[2015]= 2.486
Kučerová-Chlupáčová M., Kuneš J., Buchta V., Vejsová M., Opletalová V. 2015. Novel Pyrazine Analogs of Chalcones: Synthesis and Evaluation of Their Antifungal and Antimycobacterial Activity. Molecules. 20(1):1104-17. doi: 10.3390/molecules20011104. https://doi.org/10.3390/molecules20011104 . IF[2015]= 2.465
Karabanovich, G., Roh J., Soukup O., Pávková I., Pasdiorová M., Tambor V., Stolaříková J., Vejsová M., Vávrová K., Klimešová V., Hrabálek A. 2015. Tetrazole regioisomers in the development of nitro group-containing antitubercular agents. Med. Chem. Commun. 6, 174-181. https://doi.org/10.1039/C4MD00301B . IF[2015]= 2.54